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Discovery of Potential, Dual-Active Histamine H(3) Receptor Ligands with Combined Antioxidant Properties

In an attempt to find new dual acting histamine H(3) receptor (H(3)R) ligands, we designed a series of compounds, structurally based on previously described in our group, a highly active and selective human histamine H(3) receptor (hH(3)R) ligand KSK63. As a result, 15 obtained compounds show modera...

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Detalles Bibliográficos
Autores principales:	Kuder, Kamil J., Kotańska, Magdalena, Szczepańska, Katarzyna, Mika, Kamil, Reiner-Link, David, Stark, Holger, Kieć-Kononowicz, Katarzyna
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8071534/ https://www.ncbi.nlm.nih.gov/pubmed/33921144 http://dx.doi.org/10.3390/molecules26082300

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