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Physicochemical properties and Mycobacterium tuberculosis transporters: keys to efficacious antitubercular drugs?

Securing novel, safe, and effective medicines to treat Mycobacterium tuberculosis remains an elusive goal, particularly influenced by the largely impervious Mtb envelope that limits exposure and thus efficacy of inhibitors at their cellular and periplasmic targets. The impact of physicochemical prop...

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Detalles Bibliográficos
Autores principales: Fullam, Elizabeth, Young, Robert J.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: RSC 2020
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8130550/
https://www.ncbi.nlm.nih.gov/pubmed/34041481
http://dx.doi.org/10.1039/d0md00265h

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