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Design, Synthesis, Anticancer Evaluation, Enzymatic Assays, and a Molecular Modeling Study of Novel Pyrazole–Indole Hybrids
[Image: see text] The molecular hybridization concept has recently emerged as a powerful approach in drug discovery. A series of novel indole derivatives linked to the pyrazole moiety were designed and developed via a molecular hybridization protocol as antitumor agents. The target compounds (5a–j a...
Autores principales: | Hassan, Ashraf S., Moustafa, Gaber O., Awad, Hanem M., Nossier, Eman S., Mady, Mohamed F. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2021
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8154124/ https://www.ncbi.nlm.nih.gov/pubmed/34056388 http://dx.doi.org/10.1021/acsomega.1c01604 |
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