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Lewis acid mediated, mild C–H aminoalkylation of azoles via three component coupling

This manuscript reports the development of a mild, highly functional group tolerant and metal-free C–H aminoalkylation of azoles via a three-component coupling approach. This method enables the C–H functionalization of diverse azole substrates, such as oxazoles, benzoxazoles, thiazoles, benzothiazol...

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Detalles Bibliográficos
Autores principales:	Emmert, Marion H., He, Cyndi Qixin, Shah, Akshay A., Felten, Stephanie
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2021
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8179430/ https://www.ncbi.nlm.nih.gov/pubmed/34163658 http://dx.doi.org/10.1039/d0sc06868c

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