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Rapid and Sensitive Quantification of Intracellular Glycyl-Sarcosine for Semi-High-Throughput Screening for Inhibitors of PEPT-1

The peptide transporter PEPT-1 (SLC15A1) plays a major role in nutritional supply with amino acids by mediating the intestinal influx of dipeptides and tripeptides generated during food digestion. Its role in the uptake of small bioactive peptides and various therapeutics makes it an important targe...

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Detalles Bibliográficos
Autores principales:	von Linde, Teresa, Bajraktari-Sylejmani, Gzona, Haefeli, Walter E., Burhenne, Jürgen, Weiss, Johanna, Sauter, Max
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8309108/ https://www.ncbi.nlm.nih.gov/pubmed/34371711 http://dx.doi.org/10.3390/pharmaceutics13071019

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