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2-Aryl-6-Polyfluoroalkyl-4-Pyrones as Promising R(F)-Building-Blocks: Synthesis and Application for Construction of Fluorinated Azaheterocycles

A convenient and general method for the direct synthesis of 2-aryl-6-(trifluoromethyl)-4-pyrones and 2-aryl-5-bromo-6-(trifluoromethyl)-4-pyrones has been developed on the basis of one-pot oxidative cyclization of (E)-6-aryl-1,1,1-trifluorohex-5-ene-2,4-diones via a bromination/dehydrobromination ap...

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Detalles Bibliográficos
Autores principales:	Usachev, Sergey A., Nigamatova, Diana I., Mysik, Daria K., Naumov, Nikita A., Obydennov, Dmitrii L., Sosnovskikh, Vyacheslav Y.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8347980/ https://www.ncbi.nlm.nih.gov/pubmed/34361567 http://dx.doi.org/10.3390/molecules26154415

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