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Asymmetric synthesis of pharmaceutically relevant 1-aryl-2-heteroaryl- and 1,2-diheteroarylcyclopropane-1-carboxylates

This study describes general methods for the enantioselective syntheses of pharmaceutically relevant 1-aryl-2-heteroaryl- and 1,2-diheteroarylcyclopropane-1-carboxylates through dirhodium tetracarboxylate-catalysed asymmetric cyclopropanation of vinyl heterocycles with aryl- or heteroaryldiazoacetat...

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Detalles Bibliográficos
Autores principales:	Sharland, Jack C., Wei, Bo, Hardee, David J., Hodges, Timothy R., Gong, Wei, Voight, Eric A., Davies, Huw M. L.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2021
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8386643/ https://www.ncbi.nlm.nih.gov/pubmed/34522315 http://dx.doi.org/10.1039/d1sc02474d

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