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Chiral Vicinal Diamines Derived from Mefloquine

[Image: see text] Novel 1,2-diamines based on the mefloquine scaffold prepared in enantiomerically pure forms resemble 9-amino-Cinchona alkaloids. Most effectively, 11-aminomefloquine with an erythro configuration was obtained by conversion of 11-alcohol into azide and hydrogenation. Alkylation of a...

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Detalles Bibliográficos
Autores principales:	Kucharski, Dawid J., Kowalczyk, Rafał, Boratyński, Przemysław J.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2021
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8389910/ https://www.ncbi.nlm.nih.gov/pubmed/34314190 http://dx.doi.org/10.1021/acs.joc.1c01316

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