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Novel Functionalized Amino Acids as Inhibitors of GABA Transporters with Analgesic Activity

[Image: see text] Neuropathic pain resistance to pharmacotherapy has encouraged researchers to develop effective therapies for its treatment. γ-Aminobutyric acid (GABA) transporters 1 and 4 (mGAT1 and mGAT4) have been increasingly recognized as promising drug targets for neuropathic pain (NP) associ...

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Detalles Bibliográficos
Autores principales:	Gryzło, Beata, Zaręba, Paula, Malawska, Katarzyna, Mazur, Gabriela, Rapacz, Anna, Ła̧tka, Kamil, Höfner, Georg C., Latacz, Gniewomir, Bajda, Marek, Sałat, Kinga, Wanner, Klaus T., Malawska, Barbara, Kulig, Katarzyna
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2021
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8397297/ https://www.ncbi.nlm.nih.gov/pubmed/34347423 http://dx.doi.org/10.1021/acschemneuro.1c00351

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