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Novel Sulfonamide-Based Carbamates as Selective Inhibitors of BChE

A series of 14 target benzyl [2-(arylsulfamoyl)-1-substituted-ethyl]carbamates was prepared by multi-step synthesis and characterized. All the final compounds were tested for their ability to inhibit acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) in vitro, and the selectivity index (SI...

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Detalles Bibliográficos
Autores principales:	Magar, Pratibha, Parravicini, Oscar, Štěpánková, Šárka, Svrčková, Katarina, Garro, Adriana D., Jendrzejewska, Izabela, Pauk, Karel, Hošek, Jan, Jampílek, Josef, Enriz, Ricardo D., Imramovský, Aleš
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8430704/ https://www.ncbi.nlm.nih.gov/pubmed/34502357 http://dx.doi.org/10.3390/ijms22179447

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