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Anticancer Effects of I-BET151, an Inhibitor of Bromodomain and Extra-Terminal Domain Proteins
I-BET151 is an inhibitor of bromodomain and extra-terminal domain (BET) proteins that selectively inhibits BET family members (BRD2, BRD3, BRD4, and BRDT). Over the past ten years, many studies have demonstrated the potential of I-BET151 in cancer treatment. Specifically, I-BET151 causes cell cycle...
Autores principales: | Lai, Jiacheng, Liu, Ziqiang, Zhao, Yulei, Ma, Chengyuan, Huang, Haiyan |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Frontiers Media S.A.
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8443787/ https://www.ncbi.nlm.nih.gov/pubmed/34540687 http://dx.doi.org/10.3389/fonc.2021.716830 |
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