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Asymmetric Synthesis of 2‐Arylindolines and 2,2‐Disubstituted Indolines by Kinetic Resolution
Kinetic resolution of 2‐arylindolines (2,3‐dihydroindoles) was achieved by treatment of their N‐tert‐butoxycarbonyl (Boc) derivatives with n‐butyllithium and sparteine in toluene at −78 °C followed by electrophilic quench. The unreacted starting materials together with the 2,2‐disubstituted products...
Autores principales: | Choi, Anthony, El‐Tunsi, Ashraf, Wang, Yuhang, Meijer, Anthony J. H. M., Li, Jia, Li, Xiabing, Proietti Silvestri, Ilaria, Coldham, Iain |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
John Wiley and Sons Inc.
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8456874/ https://www.ncbi.nlm.nih.gov/pubmed/34110662 http://dx.doi.org/10.1002/chem.202101248 |
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