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Asymmetric Synthesis of 2‐Arylindolines and 2,2‐Disubstituted Indolines by Kinetic Resolution

Kinetic resolution of 2‐arylindolines (2,3‐dihydroindoles) was achieved by treatment of their N‐tert‐butoxycarbonyl (Boc) derivatives with n‐butyllithium and sparteine in toluene at −78 °C followed by electrophilic quench. The unreacted starting materials together with the 2,2‐disubstituted products...

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Detalles Bibliográficos
Autores principales:	Choi, Anthony, El‐Tunsi, Ashraf, Wang, Yuhang, Meijer, Anthony J. H. M., Li, Jia, Li, Xiabing, Proietti Silvestri, Ilaria, Coldham, Iain
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	John Wiley and Sons Inc. 2021
Materias:	Full Papers
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8456874/ https://www.ncbi.nlm.nih.gov/pubmed/34110662 http://dx.doi.org/10.1002/chem.202101248

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