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Radiosynthesis of 5-[(18)F]Fluoro-1,2,3-triazoles through Aqueous Iodine–[(18)F]Fluorine Exchange Reaction

In this report, a simple and efficient process to achieve fluorine-18-labeled 1,2,3-triazole is reported. The heteroaromatic radiofluorination was successfully achieved through an iodine–fluorine-18 exchange in an aqueous medium requiring only trace amounts of base and no azeotropic drying of fluori...

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Detalles Bibliográficos
Autores principales:	Zhang, Xiang, Basuli, Falguni, Abdelwahed, Sameh, Begley, Tadhg, Swenson, Rolf
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8469629/ https://www.ncbi.nlm.nih.gov/pubmed/34576993 http://dx.doi.org/10.3390/molecules26185522

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