Cargando…

Bisphenol A derivatives act as novel coactivator-binding inhibitors for estrogen receptor β

Bisphenol A and its derivatives are recognized as endocrine disruptors based on their complex effects on estrogen receptor (ER) signaling. While the effects of bisphenol derivatives on ERα have been thoroughly evaluated, how these chemicals affect ERβ signaling is less well understood. Herein, we so...

Descripción completa

Detalles Bibliográficos
Autores principales:	Iwamoto, Masaki, Masuya, Takahiro, Hosose, Mari, Tagawa, Koki, Ishibashi, Tomoka, Suyama, Keitaro, Nose, Takeru, Yoshihara, Eiji, Downes, Michael, Evans, Ronald M., Matsushima, Ayami
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Society for Biochemistry and Molecular Biology 2021
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8551653/ https://www.ncbi.nlm.nih.gov/pubmed/34499926 http://dx.doi.org/10.1016/j.jbc.2021.101173

Ejemplares similares

High cytotoxicity of a degraded TBBPA, dibromobisphenol A, through apoptotic and necrosis pathways
por: Suyama, Keitaro, et al.
Publicado: (2023)

Bisphenol-C is the strongest bifunctional ERα-agonist and ERβ-antagonist due to magnified halogen bonding
por: Liu, Xiaohui, et al.
Publicado: (2021)

Discovery of novel oestrogen receptor α agonists and antagonists by screening a revisited privileged structure moiety for nuclear receptors
por: Masuya, Takahiro, et al.
Publicado: (2019)

Bisphenol AF Is a Full Agonist for the Estrogen Receptor ERα but a Highly Specific Antagonist for ERβ
por: Matsushima, Ayami, et al.
Publicado: (2010)

Direct Evidence Revealing Structural Elements Essential for the High Binding Ability of Bisphenol A to Human Estrogen-Related Receptor-γ
por: Okada, Hiroyuki, et al.
Publicado: (2008)

Simple Regulation of the Self-Assembling Ability by Multimerization of Elastin-Derived Peptide (FPGVG)(n) Using Nitrilotriacetic Acid as a Building Block
por: Suyama, Keitaro, et al.
Publicado: (2021)

A Characteristic Back Support Structure in the Bisphenol A-Binding Pocket in the Human Nuclear Receptor ERRγ
por: Liu, Xiaohui, et al.
Publicado: (2014)

Metal ion scavenging activity of elastin-like peptide analogues containing a cadmium ion binding sequence
por: Sumiyoshi, Shogo, et al.
Publicado: (2022)

Nuclear role for human Argonaute-1 as an estrogen-dependent transcription coactivator
por: Gómez Acuña, Luciana I., et al.
Publicado: (2020)

In Vivo Imaging of Activated Estrogen Receptors in Utero by Estrogens and Bisphenol A
por: Lemmen, Josephine G., et al.
Publicado: (2004)

Estrogen receptor independent neurotoxic mechanism of bisphenol A, an environmental estrogen
por: Lee, Yoot Mo, et al.
Publicado: (2007)

Development of truncated elastin-like peptide analogues with improved temperature-response and self-assembling properties
por: Sumiyoshi, Shogo, et al.
Publicado: (2022)

Differential Estrogenic Actions of Endocrine-Disrupting Chemicals Bisphenol A, Bisphenol AF, and Zearalenone through Estrogen Receptor α and β in Vitro
por: Li, Yin, et al.
Publicado: (2012)

Environmental estrogens induce transcriptionally active estrogen receptor dimers in yeast: activity potentiated by the coactivator RIP140.
por: Sheeler, C Q, et al.
Publicado: (2000)

Significant Association of Estrogen Receptor-β Isoforms and Coactivators in Breast Cancer Subtypes
por: Choi, Young, et al.
Publicado: (2023)

Coactivators enable glucocorticoid receptor recruitment to fine-tune estrogen receptor transcriptional responses
por: Bolt, Michael J., et al.
Publicado: (2013)

The marionette mechanism of domain–domain communication in the antagonist, agonist, and coactivator responses of the estrogen receptor
por: Chen, Xun, et al.
Publicado: (2023)

Bisphenol A in dental sealants and its estrogen like effect
por: Rathee, Manu, et al.
Publicado: (2012)

Development of a Novel Molecular Sensor for Imaging Estrogen Receptor-Coactivator Protein-Protein Interactions
por: Lake, Madryn C., et al.
Publicado: (2012)

Implications of the Estrogen Receptor Coactivators SRC1 and SRC2 in the Biological Basis of Gender Incongruence
por: Ramírez, Karla del Valle, et al.
Publicado: (2021)

Transcriptional coactivator MED1 in the interface of anti-estrogen and anti-HER2 therapeutic resistance
por: Bick, Gregory, et al.
Publicado: (2022)

The Environmental Estrogen Bisphenol A Inhibits Estradiol-Induced Hippocampal Synaptogenesis
por: MacLusky, Neil J., et al.
Publicado: (2005)

Bisphenol A Exposure Is Associated with in Vivo Estrogenic Gene Expression in Adults
por: Melzer, David, et al.
Publicado: (2011)

Gene Alterations of Ovarian Cancer Cells Expressing Estrogen Receptors by Estrogen and Bisphenol A Using Microarray Analysis
por: Hwang, Kyung-A, et al.
Publicado: (2011)

Corepressor/coactivator paradox: potential constitutive coactivation by corepressor splice variants
por: Meng, Xianwang, et al.
Publicado: (2006)

Early cerebral activities of the environmental estrogen bisphenol A appear to act via the somatostatin receptor subtype sst(2).
por: Facciolo, Rosa Maria, et al.
Publicado: (2002)

Increasing the sensitivity of the rodent uterotrophic assay to estrogens, with particular reference to bisphenol A.
por: Ashby, J
Publicado: (2001)

Biotransformation of Bisphenol AF to Its Major Glucuronide Metabolite Reduces Estrogenic Activity
por: Li, Ming, et al.
Publicado: (2013)

Estrogen-induced transcription at individual alleles is independent of receptor level and active conformation but can be modulated by coactivators activity
por: Stossi, Fabio, et al.
Publicado: (2020)

The mouse uterotrophic assay: a reevaluation of its validity in assessing the estrogenicity of bisphenol A.
por: Markey, C M, et al.
Publicado: (2001)

In vitro estrogenicity of polybrominated diphenyl ethers, hydroxylated PDBEs, and polybrominated bisphenol A compounds.
por: Meerts, I A, et al.
Publicado: (2001)

The estrogenicity of bisphenol A-related diphenylalkanes with various substituents at the central carbon and the hydroxy groups.
por: Perez, P, et al.
Publicado: (1998)

Experimental Data Extraction and in Silico Prediction of the Estrogenic Activity of Renewable Replacements for Bisphenol A
por: Hong, Huixiao, et al.
Publicado: (2016)

A Novel Action of Endocrine-Disrupting Chemicals on Wildlife; DDT and Its Derivatives Have Remained in the Environment
por: Matsushima, Ayami
Publicado: (2018)

Biodegradation of Bisphenol A, Bisphenol F and Bisphenol S in Seawater
por: Danzl, Erica, et al.
Publicado: (2009)

3D Models of MBP, a Biologically Active Metabolite of Bisphenol A, in Human Estrogen Receptor α and Estrogen Receptor β
por: Baker, Michael E., et al.
Publicado: (2012)

The role of coactivators in oestrogen action
por: Brown, M, et al.
Publicado: (2000)

Coactivation sign in fixed dystonia
por: Mehta, Arpan R., et al.
Publicado: (2013)

Structure of transcription coactivator SAGA
por: Wang, Haibo, et al.
Publicado: (2020)

Coactivation of estrogen receptor alpha by the DEAD-box RNA helicases p68 and p72 and its role in breast cancer
por: Fuller-Pace, FV, et al.
Publicado: (2008)

Cannot write session to /tmp/vufind_sessions/sess_rh4ciuf67rsgb08qnug14rucst