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Synthesis of new bile acid-fused tetrazoles using the Schmidt reaction

A practical and high-yielding Schmidt reaction for the synthesis of fused tetrazoles from bile acid precursors was developed. Mild reaction conditions using TMSN(3) instead of hydrazoic acid as an azide source produced good yields of the desired tetrazoles. These conditions could be applied to other...

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Detalles Bibliográficos
Autores principales:	Škorić, Dušan Đ, Klisurić, Olivera R, Jakimov, Dimitar S, Sakač, Marija N, Csanádi, János J
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2021
Materias:	Full Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8551880/ https://www.ncbi.nlm.nih.gov/pubmed/34760027 http://dx.doi.org/10.3762/bjoc.17.174

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