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New Antagonists of the Membrane Androgen Receptor OXER1 from the ZINC Natural Product Database
[Image: see text] OXER1 (oxoeicosanoid receptor 1) was deorphanized in 1993 and found to be the specific receptor for the arachidonic acid metabolite 5-oxo-ETE. Recently, we have reported that androgen binds to this receptor also, being a membrane androgen receptor, triggering a number of its membra...
Autores principales: | Panagiotopoulos, Athanasios A., Kalyvianaki, Konstantina, Notas, George, Pirintsos, Stergios A., Castanas, Elias, Kampa, Marilena |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2021
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8582029/ https://www.ncbi.nlm.nih.gov/pubmed/34778638 http://dx.doi.org/10.1021/acsomega.1c04027 |
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