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Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases
Pim kinases (proviral integration site for Moloney murine leukemia virus kinases) are overexpressed in various types of hematological malignancies and solid carcinomas, and promote cell proliferation and survival. Thus, Pim kinases are validated as targets for antitumor therapy. In this context, our...
Autores principales: | Dao, Viet Hung, Ourliac-Garnier, Isabelle, Logé, Cédric, McCarthy, Florence O., Bach, Stéphane, da Silva, Teresinha Gonçalves, Denevault-Sabourin, Caroline, Thiéfaine, Jérôme, Baratte, Blandine, Robert, Thomas, Gouilleux, Fabrice, Brachet-Botineau, Marie, Bazin, Marc-Antoine, Marchand, Pascal |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8587151/ https://www.ncbi.nlm.nih.gov/pubmed/34770981 http://dx.doi.org/10.3390/molecules26216572 |
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