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Solid-Phase Synthesis of Selectively Mono-Fluorobenz(o)ylated Polyamines as a Basis for the Development of (18)F-Labeled Radiotracers

Polyamines are highly attractive vectors for tumor targeting, particularly with regards to the development of radiolabeled probes for imaging by positron emission (PET) and single-photon emission computed tomography (SPECT). However, the synthesis of selectively functionalized derivatives remains ch...

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Detalles Bibliográficos
Autores principales:	Wodtke, Robert, Pietzsch, Jens, Löser, Reik
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8625420/ https://www.ncbi.nlm.nih.gov/pubmed/34834103 http://dx.doi.org/10.3390/molecules26227012

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