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Application of QSAR Method in the Design of Enhanced Antimalarial Derivatives of Azetidine-2-carbonitriles, their Molecular Docking, Drug-likeness, and SwissADME Properties
The resistance of the P. falciparum strain to some of the antimalarial drugs has been a dominant dilemma facing the treatment of this fetid disease. This necessitates the detection and development of new antimalarial agents targeting the P. falciparum. Azetidine-2-carbonitriles reported for its anti...
Autores principales: | Ibrahim, Zakari Ya’u, Uzairu, Adamu, Shallangwa, Gideon Adamu, Abechi, Stephen Eyije |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Shaheed Beheshti University of Medical Sciences
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8653669/ https://www.ncbi.nlm.nih.gov/pubmed/34903987 http://dx.doi.org/10.22037/ijpr.2021.114536.14901 |
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