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The discovery of a novel series of potential ERRα inverse agonists based on p-nitrobenzenesulfonamide template for triple-negative breast cancer in vivo
Oestrogen related receptor α participated in the regulation of oxidative metabolism and mitochondrial biogenesis, and was overexpressed in many cancers including triple-negative breast cancer. A set of new ERRα inverse agonists based on p-nitrobenzenesulfonamide template were discovered and compound...
Autores principales: | Gao, Zhipei, Wang, Tianxiao, Li, Rui, Du, Yongli, Lv, Han, Zhang, Liudi, Chen, Haifei, Shi, Xiaojin, Li, Qunyi, Shen, Jingkang |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Taylor & Francis
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8667933/ https://www.ncbi.nlm.nih.gov/pubmed/34894977 http://dx.doi.org/10.1080/14756366.2021.1995728 |
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