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In Vitro and In Silico Characterization of Kurarinone as a Dopamine D(1A) Receptor Antagonist and D(2L) and D(4) Receptor Agonist

[Image: see text] Alterations in the expression and/or activity of brain G-protein-coupled receptors (GPCRs) such as dopamine D(1)R, D(2L)R, D(3)R, and D(4)R, vasopressin V(1A)R, and serotonin 5-HT(1A)R are noted in various neurodegenerative diseases (NDDs). Since studies have indicated that flavono...

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Detalles Bibliográficos
Autores principales: Prajapati, Ritu, Seong, Su Hui, Paudel, Pradeep, Park, Se Eun, Jung, Hyun Ah, Choi, Jae Sue
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2021
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8674921/
https://www.ncbi.nlm.nih.gov/pubmed/34926894
http://dx.doi.org/10.1021/acsomega.1c04109

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