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In Vitro and In Silico Characterization of Kurarinone as a Dopamine D(1A) Receptor Antagonist and D(2L) and D(4) Receptor Agonist
[Image: see text] Alterations in the expression and/or activity of brain G-protein-coupled receptors (GPCRs) such as dopamine D(1)R, D(2L)R, D(3)R, and D(4)R, vasopressin V(1A)R, and serotonin 5-HT(1A)R are noted in various neurodegenerative diseases (NDDs). Since studies have indicated that flavono...
Autores principales: | Prajapati, Ritu, Seong, Su Hui, Paudel, Pradeep, Park, Se Eun, Jung, Hyun Ah, Choi, Jae Sue |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2021
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8674921/ https://www.ncbi.nlm.nih.gov/pubmed/34926894 http://dx.doi.org/10.1021/acsomega.1c04109 |
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