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New Heterocyclic Combretastatin A-4 Analogs: Synthesis and Biological Activity of Styryl-2(3H)-benzothiazolones

Here, we describe the synthesis, characterization, and biological activities of a series of 26 new styryl-2(3H)-benzothiazolone analogs of combretastatin-A4 (CA-4). The cytotoxic activities of these compounds were tested in several cell lines (EA.hy926, A549, BEAS-2B, MDA-MB-231, HT-29, MCF-7, and M...

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Detalles Bibliográficos
Autores principales: Atanasov, Gjorgji, Rusew, Rusi I., Gelev, Vladimir M., Chanev, Christo D., Nikolova, Rosica, Shivachev, Boris L., Petrov, Ognyan I., Apostolova, Margarita D.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2021
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8703450/
https://www.ncbi.nlm.nih.gov/pubmed/34959731
http://dx.doi.org/10.3390/ph14121331

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