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Distinct In Vitro Binding Profile of the Somatostatin Receptor Subtype 2 Antagonist [(177)Lu]Lu-OPS201 Compared to the Agonist [(177)Lu]Lu-DOTA-TATE

Treatment of neuroendocrine tumours with the radiolabelled somatostatin receptor subtype 2 (SST(2)) peptide agonist [(177)Lu]Lu-DOTA-TATE is effective and well-established. Recent studies suggest improved therapeutic efficacy using the SST(2) peptide antagonist [(177)Lu]Lu-OPS201. However, little is...

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Detalles Bibliográficos
Autores principales:	Mansi, Rosalba, Plas, Pascale, Vauquelin, Georges, Fani, Melpomeni
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2021
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8706879/ https://www.ncbi.nlm.nih.gov/pubmed/34959665 http://dx.doi.org/10.3390/ph14121265

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