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High-Throughput Screening Campaign Identified a Potential Small Molecule RXFP3/4 Agonist
Relaxin/insulin-like family peptide receptor 3 (RXFP3) belongs to class A G protein-coupled receptor family. RXFP3 and its endogenous ligand relaxin-3 are mainly expressed in the brain with important roles in the regulation of appetite, energy metabolism, endocrine homeostasis and emotional processi...
Autores principales: | Lin, Guangyao, Feng, Yang, Cai, Xiaoqing, Zhou, Caihong, Shao, Lijun, Chen, Yan, Chen, Linhai, Liu, Qing, Zhou, Qingtong, Bathgate, Ross A.D., Yang, Dehua, Wang, Ming-Wei |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8709172/ https://www.ncbi.nlm.nih.gov/pubmed/34946593 http://dx.doi.org/10.3390/molecules26247511 |
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