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Acid-Catalyzed Hydrolysis and Intramolecular Cyclization of N-Cyano Sulfoximines for the Synthesis of Thiadiazine 1-Oxides

[Image: see text] Herein, we describe a novel approach for the practical synthesis of thiadiazine 1-oxides 10. The first example of an intramolecular cyclization with 2-N-cyano-sulfonimidoyl amides 9 to form the desired thiadiazine 1-oxides 10 was developed. One-pot acid-induced hydrolysis of the cy...

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Detalles Bibliográficos
Autores principales:	Oh, In Seok, Seo, Ye Ji, Hyun, Ji Young, Lim, Hwan Jung, Lee, Duck-Hyung, Park, Seong Jun
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2022
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8771986/ https://www.ncbi.nlm.nih.gov/pubmed/35071904 http://dx.doi.org/10.1021/acsomega.1c05570

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