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Disrupting GPCR Complexes with Smart Drug-like Peptides

G protein-coupled receptors (GPCRs) are a superfamily of proteins classically described as monomeric transmembrane (TM) receptors. However, increasing evidence indicates that many GPCRs form higher-order assemblies made up of monomers pertaining to identical (homo) or to various (hetero) receptors....

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Detalles Bibliográficos
Autores principales: Gallo, Maria, Defaus, Sira, Andreu, David
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8779866/
https://www.ncbi.nlm.nih.gov/pubmed/35057055
http://dx.doi.org/10.3390/pharmaceutics14010161