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Impact of the mouse model and molar amount of injected ligand on the tissue distribution profile of PSMA radioligands

PURPOSE: Various preclinical study designs are described in the literature for the evaluation of PSMA radioligands. In this study, [(177)Lu]Lu-Ibu-DAB-PSMA, an albumin-binding radioligand, and [(177)Lu]Lu-PSMA-617 were investigated and compared under variable experimental conditions. METHODS: In vit...

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Detalles Bibliográficos
Autores principales: Tschan, Viviane J., Borgna, Francesca, Schibli, Roger, Müller, Cristina
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Springer Berlin Heidelberg 2021
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8803738/
https://www.ncbi.nlm.nih.gov/pubmed/34402925
http://dx.doi.org/10.1007/s00259-021-05446-5