Cargando…
In Vitro Biological Evaluation of Aprepitant Based (177)Lu-Radioconjugates
Currently, the search for promising NK1R-positive tumor-targeting radiopharmaceuticals based on the structure of small molecular antagonists of neurokinin-1 receptor can be observed. Following this trend, we continued our evaluation of aprepitant-based (177)Lu-radioconjugates in terms of future onco...
Autores principales: | Halik, Paweł K., Koźmiński, Przemysław, Matalińska, Joanna, Lipiński, Piotr F. J., Misicka, Aleksandra, Gniazdowska, Ewa |
---|---|
Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2022
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8949964/ https://www.ncbi.nlm.nih.gov/pubmed/35335981 http://dx.doi.org/10.3390/pharmaceutics14030607 |
Ejemplares similares
-
Radiochemical Synthesis and Evaluation of Novel Radioconjugates of Neurokinin 1 Receptor Antagonist Aprepitant Dedicated for NK1R-Positive Tumors
por: Halik, Paweł K., et al.
Publicado: (2020) -
Novel NK1R-Targeted (68)Ga-/(177)Lu-Radioconjugates with Potential Application against Glioblastoma Multiforme: Preliminary Exploration of Structure–Activity Relationships
por: Matalińska, Joanna, et al.
Publicado: (2022) -
Synthesis, Physicochemical and Biological Study of Gallium-68- and Lutetium-177-Labeled VEGF-A(165)/NRP-1 Complex Inhibitors Based on Peptide A7R and Branched Peptidomimetic
por: Masłowska, Katarzyna, et al.
Publicado: (2022) -
Perspectives of Methotrexate-Based Radioagents for
Application in Nuclear Medicine
por: Halik, Paweł Krzysztof, et al.
Publicado: (2020) -
Overview of Dual-Acting Drug Methotrexate in Different Neurological Diseases, Autoimmune Pathologies and Cancers
por: Koźmiński, Przemysław, et al.
Publicado: (2020)