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Beta and Gamma Amino Acid-Substituted Benzenesulfonamides as Inhibitors of Human Carbonic Anhydrases

A series of novel benzenesulfonamide derivatives were synthesized bearing para-N β,γ-amino acid or para-N β-amino acid and thiazole moieties and their binding to the human carbonic anhydrase (CA) isozymes determined. These enzymes are involved in various illnesses, such as glaucoma, altitude sicknes...

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Detalles Bibliográficos
Autores principales:	Balandis, Benas, Šimkūnas, Tomas, Paketurytė-Latvė, Vaida, Michailovienė, Vilma, Mickevičiūtė, Aurelija, Manakova, Elena, Gražulis, Saulius, Belyakov, Sergey, Kairys, Visvaldas, Mickevičius, Vytautas, Zubrienė, Asta, Matulis, Daumantas
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9033141/ https://www.ncbi.nlm.nih.gov/pubmed/35455474 http://dx.doi.org/10.3390/ph15040477

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