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Development of structurally extended benzosiloxaboroles – synthesis and in vitro biological evaluation

The synthesis of potassium 6-hydroxy-7-chloro-1,1-dimethyl-3,3-difluorobenzo-1,2,3-siloxaborolate 5b from readily available 4-bromo-2-chlorophenol was developed. This compound proved useful in various derivatizations resulting in a wide range of O-functionalized benzosiloxaboroles. Reactions of 5b w...

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Detalles Bibliográficos
Autores principales:	Pacholak, P., Krajewska, J., Wińska, P., Dunikowska, J., Gogowska, U., Mierzejewska, J., Durka, K., Woźniak, K., Laudy, A. E., Luliński, S.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2021
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9037100/ https://www.ncbi.nlm.nih.gov/pubmed/35478884 http://dx.doi.org/10.1039/d1ra04127d

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