Cargando…

Emergent antibacterial activity of N-(thiazol-2-yl)benzenesulfonamides in conjunction with cell-penetrating octaarginine

Hybrid antimicrobials that combine the effect of two or more agents represent a promising antibacterial therapeutic strategy. In this work, we have synthesized N-(4-(4-(methylsulfonyl)phenyl)-5-phenylthiazol-2-yl)benzenesulfonamide derivatives that combine thiazole and sulfonamide, groups with known...

Descripción completa

Detalles Bibliográficos
Autores principales:	Ratrey, Poonam, Das Mahapatra, Amarjyoti, Pandit, Shiny, Hadianawala, Murtuza, Majhi, Sasmita, Mishra, Abhijit, Datta, Bhaskar
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2021
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9038147/ https://www.ncbi.nlm.nih.gov/pubmed/35478531 http://dx.doi.org/10.1039/d1ra03882f

Ejemplares similares

Enhancing Aqueous Solubility and Antibacterial Activity of Curcumin by Complexing with Cell-Penetrating Octaarginine
por: Ratrey, Poonam, et al.
Publicado: (2020)

The Effect of Conjugation with Octaarginine, a Cell-Penetrating Peptide on Antifungal Activity of Imidazoacridinone Derivative
por: Rząd, Kamila, et al.
Publicado: (2021)

Small Molecule Soluble Epoxide Hydrolase Inhibitors in Multitarget and Combination Therapies for Inflammation and Cancer
por: Das Mahapatra, Amarjyoti, et al.
Publicado: (2020)

Octaarginine Improves the Efficacy of Nitazoxanide against Cryptosporidium parvum
por: Nguyen-Ho-Bao, Tran, et al.
Publicado: (2022)

Solid lipid nanoparticles modified with stearic acid–octaarginine for oral administration of insulin
por: Zhang, Zhen-Hai, et al.
Publicado: (2012)

Live‐cell imaging of octaarginine‐modified polymer dots via single particle tracking
por: Luo, Yao, et al.
Publicado: (2019)

Cooperative Cellular Uptake and Activity of Octaarginine Antisense Peptide Nucleic Acid (PNA) Conjugates
por: Ghavami, Mahdi, et al.
Publicado: (2019)

Octaarginine-modified gold nanoparticles enhance the radiosensitivity of human colorectal cancer cell line LS180 to megavoltage radiation
por: Zhang, Xuyang, et al.
Publicado: (2018)

Glycosaminoglycan Binding and Non-Endocytic Membrane Translocation of Cell-Permeable Octaarginine Monitored by Real-Time In-Cell NMR Spectroscopy
por: Takechi-Haraya, Yuki, et al.
Publicado: (2017)

Unilateral conjunctivitis of unique etiology: A case report from Eastern India
por: Pal, Nandita, et al.
Publicado: (2016)

N-(2,3-Dihydro-1,3-thiazol-2-ylidene)-4-[(2-hydroxybenzylidene)amino]benzenesulfonamide
por: Zhang, Xin-Li
Publicado: (2009)

Transferrin and octaarginine modified dual-functional liposomes with improved cancer cell targeting and enhanced intracellular delivery for the treatment of ovarian cancer
por: Deshpande, Pranali, et al.
Publicado: (2018)

Evaluation of a d-Octaarginine-linked polymer as a transfection tool for transient and stable transgene expression in human and murine cell lines
por: SAKUMA, Saki, et al.
Publicado: (2022)

Design and Development of Novel Urea, Sulfonyltriurea, and Sulfonamide Derivatives as Potential Inhibitors of Sphingosine Kinase 1
por: Roy, Sonam, et al.
Publicado: (2020)

Antibacterial activity evaluation and mode of action study of novel thiazole-quinolinium derivatives
por: Li, Ying, et al.
Publicado: (2020)

Tail-approach based design, synthesis, and cytotoxic evaluation of novel disubstituted and trisubstituted 1,3-thiazole benzenesulfonamide derivatives with suggested carbonic anhydrase IX inhibition mechanism
por: Bondock, Samir, et al.
Publicado: (2023)

Thiazole Antibiotic Thiostrepton Synergize with Bortezomib to Induce Apoptosis in Cancer Cells
por: Pandit, Bulbul, et al.
Publicado: (2011)

Effective photo-enhancement of cellular activity of fluorophore-octaarginine antisense PNA conjugates correlates with singlet oxygen formation, endosomal escape and chromophore lipophilicity
por: Yarani, Reza, et al.
Publicado: (2018)

4-Methyl-N-(4-methylphenylsulfonyl)-N-[4-(4-methylphenyl)-1,3-thiazol-2-yl]benzenesulfonamide
por: Carballo, Rubén M., et al.
Publicado: (2013)

Antibacterial Characterization of Novel Synthetic Thiazole Compounds against Methicillin-Resistant Staphylococcus pseudintermedius
por: Mohammad, Haroon, et al.
Publicado: (2015)

Antibacterial activity of 3-methylbenzo[d]thiazol-methylquinolinium derivatives and study of their action mechanism
por: Sun, Ning, et al.
Publicado: (2018)

4-(Benzylideneamino)benzenesulfonamide
por: Loughrey, Bradley T., et al.
Publicado: (2009)

Synthesis and Antidiabetic Evaluation of Benzenesulfonamide Derivatives
por: Hosseinzadeh, Nouraddin, et al.
Publicado: (2013)

Integrated analysis of three bacterial conjunctivitis trials of besifloxacin ophthalmic suspension, 0.6%: etiology of bacterial conjunctivitis and antibacterial susceptibility profile
por: Haas, Wolfgang, et al.
Publicado: (2011)

Simulation-Optimization for Conjunctive Water Resources Management and Optimal Crop Planning in Kushabhadra-Bhargavi River Delta of Eastern India
por: Jha, Madan K., et al.
Publicado: (2020)

Synthesis and in vitro antibacterial, antifungal, anti-proliferative activities of novel adamantane-containing thiazole compounds
por: Warda, Eman T., et al.
Publicado: (2022)

N-(1-Naphthyl)benzenesulfonamide
por: Zhang, Sifang, et al.
Publicado: (2011)

A Thiazole Orange Derivative Targeting the Bacterial Protein FtsZ Shows Potent Antibacterial Activity
por: Sun, Ning, et al.
Publicado: (2017)

Conjunctivitis
Publicado: (1907)

Treatment of Conjunctivitis: II. Purulent and Gonorrhœal Conjunctivitis
Publicado: (1907)

Cell penetrating thiazole peptides inhibit c-MYC expression via site-specific targeting of c-MYC G-quadruplex
por: Dutta, Debasish, et al.
Publicado: (2018)

Synthesis, antibacterial and antioxidant activities of Thiazole-based Schiff base derivatives: a combined experimental and computational study
por: Lemilemu, Fitsum, et al.
Publicado: (2021)

A green synthesis and antibacterial activity of ferrocene-based thiazole derivatives in choline chloride/glycerol eutectic solvent
por: Zhao, Di, et al.
Publicado: (2022)

A Novel Strategy for the Design of Aurein 1.2 Analogs with Enhanced Bioactivities by Conjunction of Cell-Penetrating Regions
por: Liao, Fengting, et al.
Publicado: (2023)

2-Nitro-N-(4-pyridinio)benzenesulfonamidate
por: Li, Jiang-Sheng, et al.
Publicado: (2007)

N-(2-Methylphenyl)benzenesulfonamide
por: Gowda, B. Thimme, et al.
Publicado: (2008)

N-(3-Methylbenzoyl)benzenesulfonamide
por: Suchetan, P. A., et al.
Publicado: (2012)

N-(3-Nitrobenzoyl)benzenesulfonamide
por: Suchetan, P. A., et al.
Publicado: (2012)

N-Acetyl-4-(benzenesulfonamido)benzenesulfonamide
por: Ashfaq, Muhammad, et al.
Publicado: (2009)

N-(2-Chlorobenzoyl)benzenesulfonamide
por: Gowda, B. Thimme, et al.
Publicado: (2010)

Cannot write session to /tmp/vufind_sessions/sess_84iqnmvd8qu7begilg3j4pb7l6