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A mild and concise synthesis of aryloxy phosphoramidate prodrug of alcohols via transesterification reaction

A synthesis of aryloxy phosphoramidate prodrug of alcohols enabled by a transesterification strategy is described here. This reaction operates under mild conditions and thus has excellent functional group tolerance. This method provides an efficient and practical solution to the rapid construction o...

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Detalles Bibliográficos
Autores principales:	Ying, Hanglu, Yao, Jie, Wu, Fan, Zhao, Yufen, Ni, Feng
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2022
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9052952/ https://www.ncbi.nlm.nih.gov/pubmed/35497010 http://dx.doi.org/10.1039/d2ra01995g

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