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An efficient 3-acylquinoline synthesis from acetophenones and anthranil via C(sp(3))–H bond activation mediated by Selectfluor

An efficient method for the synthesis of 3-functionalized quinolines from commercially available acetophenones and anthranil has been described. Selectfluor propels the C(sp(3))–H bond activation of the acetophenones and aza-Michael addition of anthranil resulting in annulated 3-acylquinolines in mo...

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Detalles Bibliográficos
Autores principales:	Gao, Yejun, Hider, Robert C., Ma, Yongmin
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2019
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9062302/ https://www.ncbi.nlm.nih.gov/pubmed/35520934 http://dx.doi.org/10.1039/c9ra01481k

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