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A solid-phase approach for the synthesis of α-aminoboronic acid peptides

A solid-phase synthesis of α-aminoboronic acid peptides using a 1-glycerol polystyrene resin is described. Standard Fmoc solid-phase peptide chemistry is carried out to construct bortezomib and ixazomib. This approach eliminates the need for liquid–liquid extractions, silica gel column chromatograph...

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Detalles Bibliográficos
Autores principales:	Daniels, Blake E., Stivala, Craig E.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2018
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9077542/ https://www.ncbi.nlm.nih.gov/pubmed/35541192 http://dx.doi.org/10.1039/c7ra13479g

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