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Novel 2-(5-Aryl-4,5-Dihydropyrazol-1-yl)thiazol-4-One as EGFR Inhibitors: Synthesis, Biological Assessment and Molecular Docking Insights

INTRODUCTION: Epidermal growth factor receptor (EGFR) regulates several cell functions which include cell growth, survival, multiplication, differentiation, and apoptosis. Currently, EGFR kinase inhibitors are of increasing interest as promising targeted antitumor therapeutic agents. METHODS: Differ...

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Detalles Bibliográficos
Autores principales: Al-Warhi, Tarfah, El Kerdawy, Ahmed M, Said, Mohamed A, Albohy, Amgad, Elsayed, Zainab M, Aljaeed, Nada, Elkaeed, Eslam B, Eldehna, Wagdy M, Abdel-Aziz, Hatem A, Abdelmoaz, Miral A
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Dove 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9123247/
https://www.ncbi.nlm.nih.gov/pubmed/35607598
http://dx.doi.org/10.2147/DDDT.S356988