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Influence of Open Chain and Cyclic Structure of Peptidomimetics on Antibacterial Activity in E. coli Strains

An efficient method for the synthesis of functionalized peptidomimetics via multicomponent Ugi reaction has been developed. The application of trifluoroethanol (TFE) as a reaction medium provided desired products with good yields. Further, using the developed cyclisation reaction, the obtained pepti...

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Detalles Bibliográficos
Autores principales:	Sahrawat, Parul, Kowalczyk, Paweł, Koszelewski, Dominik, Szymczak, Mateusz, Kramkowski, Karol, Wypych, Aleksandra, Ostaszewski, Ryszard
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9182016/ https://www.ncbi.nlm.nih.gov/pubmed/35684570 http://dx.doi.org/10.3390/molecules27113633

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