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Relationship between Structure and Antibacterial Activity of α-Aminophosphonate Derivatives Obtained via Lipase-Catalyzed Kabachnik−Fields Reaction

We reported a new method dealing with the synthesis of novel pharmacologically relevant α-aminophosphonate derivatives via a lipase-catalyzed Kabachnik−Fields reaction with yields of up to 93%. The advantages of this protocol are excellent yields, mild reaction conditions, low costs, and sustainabil...

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Detalles Bibliográficos
Autores principales:	Koszelewski, Dominik, Kowalczyk, Paweł, Śmigielski, Paweł, Samsonowicz-Górski, Jan, Kramkowski, Karol, Wypych, Aleksandra, Szymczak, Mateusz, Ostaszewski, Ryszard
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9182137/ https://www.ncbi.nlm.nih.gov/pubmed/35683150 http://dx.doi.org/10.3390/ma15113846

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