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Recent Molecular Insights into Agonist-specific Binding to the Mu-Opioid Receptor

Opioid agonists produce their analgesic effects primarily by acting at the µ-opioid receptor (µOR). µOR agonists with different efficacies exert diverse molecular changes in the µOR which dictate the faith of the receptor’s signaling pathway and possibly it’s the degree of desensitization. Since the...

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Detalles Bibliográficos
Autores principales:	Zádor, Ferenc, Király, Kornél, Essmat, Nariman, Al-Khrasani, Mahmoud
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Frontiers Media S.A. 2022
Materias:	Molecular Biosciences
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9234319/ https://www.ncbi.nlm.nih.gov/pubmed/35769909 http://dx.doi.org/10.3389/fmolb.2022.900547

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