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Exploring the kinetic selectivity of drugs targeting the β(1)‐adrenoceptor
In this study, we report the β(1)‐adrenoceptor binding kinetics of several clinically relevant β(1/2)‐adrenoceptor (β(1/2)AR) agonists and antagonists. [(3)H]‐DHA was used to label CHO‐β(1)AR for binding studies. The kinetics of ligand binding was assessed using a competition association binding met...
| Autores principales: | , , , , , |
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| Formato: | Online Artículo Texto |
| Lenguaje: | English |
| Publicado: |
John Wiley and Sons Inc.
2022
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| Materias: | |
| Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9237807/ https://www.ncbi.nlm.nih.gov/pubmed/35762357 http://dx.doi.org/10.1002/prp2.978 |