Cargando…
CYP11A1-derived vitamin D hydroxyderivatives as candidates for therapy of basal and squamous cell carcinomas
Hydroxyderivatives of vitamin D3, including classical 1,25(OH)(2)D3 and novel CYP11A1-derived hydroxyderivatives, exert their biological activity by acting as agonists on the vitamin D receptor (VDR) and inverse agonists on retinoid-related orphan receptors (ROR)α and γ. The anti-cancer activities o...
Autores principales: | Slominski, Andrzej T., Brożyna, Anna A., Kim, Tae-Kang, Elsayed, Mahmoud M., Janjetovic, Zorica, Qayyum, Shariq, Slominski, Radomir M., Oak, Allen S.W., Li, Changzhao, Podgorska, Ewa, Li, Wei, Jetten, Anton M., Tuckey, Robert C., Tang, Edith K.Y., Elmets, Craig, Athar, Mohammad |
---|---|
Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
D.A. Spandidos
2022
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9262157/ https://www.ncbi.nlm.nih.gov/pubmed/35775377 http://dx.doi.org/10.3892/ijo.2022.5386 |
Ejemplares similares
-
RF15 | PMON293 Metabolic activation of tachysterol to biologically active hydroxyderivatives that act on VDR, AhR, LXRs and PPARγ receptors
por: Slominski, Andrzej, et al.
Publicado: (2022) -
Knocking out the Vitamin D Receptor Enhances Malignancy and Decreases Responsiveness to Vitamin D3 Hydroxyderivatives in Human Melanoma Cells
por: Podgorska, Ewa, et al.
Publicado: (2021) -
Association among Vitamin D, Retinoic Acid-Related Orphan Receptors, and Vitamin D Hydroxyderivatives in Ovarian Cancer
por: Brożyna, Anna A., et al.
Publicado: (2020) -
CYP24A1 Expression Inversely Correlates with Melanoma Progression: Clinic-Pathological Studies
por: Brożyna, Anna A., et al.
Publicado: (2014) -
Novel CYP11A1-Derived Vitamin D and Lumisterol Biometabolites for the Management of COVID-19
por: Qayyum, Shariq, et al.
Publicado: (2022)