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Phenylboronic Ester-Activated Aryl Iodide-Selective Buchwald–Hartwig-Type Amination toward Bioactivity Assay

[Image: see text] In this study, a phenylboronic ester-activated aryl iodide-selective Buchwald–Hartwig-type amination was developed. When the reaction of aryl iodides and aryl/aliphatic amines using Ni(acac)(2) is carried out in the presence of phenylboronic ester, the Buchwald–Hartwig-type aminati...

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Detalles Bibliográficos
Autores principales:	Dhital, Raghu N., Sen, Abhijit, Hu, Hao, Ishii, Rikako, Sato, Takuma, Yashiroda, Yoko, Kimura, Hiromi, Boone, Charles, Yoshida, Minoru, Futamura, Yushi, Hirano, Hiroyuki, Osada, Hiroyuki, Hashizume, Daisuke, Uozumi, Yasuhiro, Yamada, Yoichi M.A.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2022
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9301730/ https://www.ncbi.nlm.nih.gov/pubmed/35874269 http://dx.doi.org/10.1021/acsomega.2c01092

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