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A Modular Synthesis of Teraryl‐Based α‐Helix Mimetics, Part 5: A Complete Set of Pyridine Boronic Acid Pinacol Esters Featuring Side Chains of Proteinogenic Amino Acids

Teraryl‐based α‐helix mimetics have proven to be useful compounds for the inhibition of protein‐protein interactions (PPI). We have developed a modular and flexible approach for the synthesis of teraryl‐based α‐helix mimetics using pyridine containing boronic acid building blocks to increase the wat...

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Detalles Bibliográficos
Autores principales:	Trobe, Melanie, Schreiner, Till, Vareka, Martin, Grimm, Sebastian, Wölfl, Bernhard, Breinbauer, Rolf
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	John Wiley and Sons Inc. 2022
Materias:	Research Articles
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9304165/ https://www.ncbi.nlm.nih.gov/pubmed/35910461 http://dx.doi.org/10.1002/ejoc.202101280

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