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New Insight into Dearomatization and Decarbonylation of Antitubercular 4H‐Benzo[e][1,3]thiazinones: Stable 5H‐ and 7H‐Benzo[e][1,3]thiazines

8‐Nitro‐4H‐benzo[e][1,3]thiazinones (BTZs) are potent in vitro antimycobacterial agents. New chemical transformations, viz. dearomatization and decarbonylation, of two BTZs and their influence on the compounds’ antimycobacterial properties are described. Reactions of 8‐nitro‐2‐(piperidin‐1‐yl)‐6‐(tr...

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Detalles Bibliográficos
Autores principales:	Richter, Adrian, Seidel, Rüdiger W., Graf, Jürgen, Goddard, Richard, Lehmann, Christoph, Schlegel, Tom, Khater, Nour, Imming, Peter
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	John Wiley and Sons Inc. 2022
Materias:	Research Articles
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9306624/ https://www.ncbi.nlm.nih.gov/pubmed/35170242 http://dx.doi.org/10.1002/cmdc.202200021

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