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N‐Terminal Selective C−H Azidation of Proline‐Containing Peptides: a Platform for Late‐Stage Diversification
A methodology for the C−H azidation of N‐terminal proline‐containing peptides was developed employing only commercially available reagents. Peptides bearing a broad range of functionalities and containing up to 6 amino acids were selectively azidated at the carbamate‐protected N‐terminal residue in...
Autores principales: | Allouche, Emmanuelle M. D., Simonet‐Davin, Raphaël, Waser, Jerome |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
John Wiley and Sons Inc.
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9306896/ https://www.ncbi.nlm.nih.gov/pubmed/35137991 http://dx.doi.org/10.1002/chem.202200368 |
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