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One-Pot Diastereoselective Synthesis of Pyrrolopiperazine-2,6-diones by a Ugi/Nucleophilic Substitution/N-Acylation Sequence

[Image: see text] The diastereoselective synthesis of two families of pyrrolopiperazine-2,6-diones is presented. These compounds were prepared by one-pot Ugi/nucleophilic substitution/N-acylation/debenzoylation/(elimination) sequences. This novel route provides straightforward access to a wide varie...

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Detalles Bibliográficos
Autores principales:	González-Saiz, Beatriz, Carreira-Barral, Israel, Pertejo, Pablo, Gómez-Ayuso, Javier, Quesada, Roberto, García-Valverde, María
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2022
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9348836/ https://www.ncbi.nlm.nih.gov/pubmed/35759645 http://dx.doi.org/10.1021/acs.joc.2c00694

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