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Discovery of the First Highly Selective Antagonist of the GluK3 Kainate Receptor Subtype

Kainate receptors belong to the family of glutamate receptors ion channels, which are responsible for the majority of rapid excitatory synaptic transmission in the central nervous system. The therapeutic potential of kainate receptors is still poorly understood, which is also due to the lack of pote...

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Detalles Bibliográficos
Autores principales:	Chałupnik, Paulina, Vialko, Alina, Pickering, Darryl S., Hinkkanen, Markus, Donbosco, Stephanie, Møller, Thor C., Jensen, Anders A., Nielsen, Birgitte, Bay, Yasmin, Kristensen, Anders S., Johansen, Tommy N., Łątka, Kamil, Bajda, Marek, Szymańska, Ewa
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9369419/ https://www.ncbi.nlm.nih.gov/pubmed/35955932 http://dx.doi.org/10.3390/ijms23158797

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