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Refined Chelator Spacer Moieties Ameliorate the Pharmacokinetics of PSMA-617

Prostate-specific membrane antigen (PSMA) binding tracers are promising agents for the targeting of prostate tumors. To further optimize the clinically established radiopharmaceutical PSMA-617, novel PSMA ligands for prostate cancer endoradiotherapy were developed. A series of PSMA binding tracers t...

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Detalles Bibliográficos
Autores principales:	dos Santos, José Carlos, Schäfer, Martin, Bauder-Wüst, Ulrike, Beijer, Barbro, Eder, Matthias, Leotta, Karin, Kleist, Christian, Meyer, Jan-Philip, Dilling, Thomas R., Lewis, Jason S., Kratochwil, Clemens, Kopka, Klaus, Haberkorn, Uwe, Mier, Walter
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Frontiers Media S.A. 2022
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9396645/ https://www.ncbi.nlm.nih.gov/pubmed/36017165 http://dx.doi.org/10.3389/fchem.2022.898692

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