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Synthesis, Structure and Antileishmanial Evaluation of Endoperoxide–Pyrazole Hybrids

Leishmaniases are among the most impacting neglected tropical diseases. In attempts to repurpose antimalarial drugs or candidates, it was found that selected 1,2,4-trioxanes, 1,2,4,5-tetraoxanes, and pyrazole-containing chemotypes demonstrated activity against Leishmania parasites. This study report...

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Detalles Bibliográficos
Autores principales: Amado, Patrícia S. M., Costa, Inês C. C., Paixão, José A., Mendes, Ricardo F., Cortes, Sofia, Cristiano, Maria L. S.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9457810/
https://www.ncbi.nlm.nih.gov/pubmed/36080174
http://dx.doi.org/10.3390/molecules27175401

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