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Identification of a Partial and Selective TRPV1 Agonist CPIPC for Alleviation of Inflammatory Pain
Transient receptor potential vanilloid 1 (TRPV1) is a non-selective cation channel, predominantly expressed in a subset of peripheral sensory neurons for pain signaling. Topical application of agonist capsaicin for desensitizing TRPV1 currents has been approved for relief of chronic pain. However, t...
Autores principales: | Dong, Liying, Zhou, Qiqi, Liang, Qianqian, Qiao, Zhen, Liu, Yani, Shao, Liming, Wang, Kewei |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9457966/ https://www.ncbi.nlm.nih.gov/pubmed/36080196 http://dx.doi.org/10.3390/molecules27175428 |
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