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Synthesis and Preclinical Evaluation of (177)Lu-Labeled Radiohybrid PSMA Ligands for Endoradiotherapy of Prostate Cancer

The prostate-specific membrane antigen (PSMA)–targeted radiohybrid (rh) ligand [(177)Lu]Lu-rhPSMA-7.3 has recently been assessed in a pretherapeutic dosimetry study on prostate cancer patients. In comparison to [(177)Lu]Lu-PSMA I&T, application of [(177)Lu]Lu-rhPSMA-7.3 resulted in a significant...

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Detalles Bibliográficos
Autores principales:	Wurzer, Alexander, Kunert, Jan-Philip, Fischer, Sebastian, Felber, Veronika, Beck, Roswitha, de Rose, Francesco, D’Alessandria, Calogero, Weber, Wolfgang, Wester, Hans-Jürgen
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Society of Nuclear Medicine 2022
Materias:	Basic Science Investigation
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9536713/ https://www.ncbi.nlm.nih.gov/pubmed/35086894 http://dx.doi.org/10.2967/jnumed.121.263371

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